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- Objective:To establish a low-cost synthetic route of thymopentin. 目的:研究免疫增強劑胸腺五肽的合成路線(xiàn),以降低合成成本。
- Objective to observe the curative effect of cisplatin on malignant pleural effusion combined with thymopentin at patients. 摘要目的觀(guān)察順鉑聯(lián)合胸腺五肽治療惡性胸腔積液的療效。
- Thymopentin (TP5) has been recently evaluated as an immunotherapeutic agent for the treatment of cancer. 胸腺五肽(TP5)近來(lái)被認為是腫瘤治療的免疫治療劑。
- OBJECTIVE To investigate the preparation of thymopentin loaded oral modified-chitosan nanoparticles(Tp5-TMC-NP). 目的探討以三甲基殼聚糖為材料制備胸腺五肽納米粒的制備條件。
- Evaluation of clinical efficacy and tolerability of intravenous high dose thymopentin in advanced melanoma patients. 大劑量靜脈注射TP5在進(jìn)展性黑色素瘤患者中的臨床應用及...
- OBJECTIVE To prepare thymopentin microspheres and investigate the drug release in vitro. 目的制備胸腺五肽微球并對其體外釋放進(jìn)行考察。
- Conclusion D-amino acids substituted peptides of thymopentin had stronger immunological activity than thymopentin. 結論D-氨基酸置換的胸腺五肽類(lèi)似物對T淋巴細胞的免疫調節作用比胸腺五肽作用更強。
- Purpose To synthesize a peptide library of thymopentin with D-amino acids substituted, and to determine its effect of lymphocytic proliferation. 摘要目的合成胸腺五肽D型氨基酸取代肽庫,并測定對T淋巴細胞的免疫活性。
- Teabag method was used to synthesize the peptide library of thymopentin with D-amino acids substituted by solid phase peptide synthesis (SPPS). 利用組合化學(xué)技術(shù),采用簡(jiǎn)便的茶袋法固相合成制備胸腺五肽D型氨基酸取代類(lèi)似物肽庫,共合成32條肽。
- There are some surely therapeutic effect for cisplatin combination with thymopentin on patients with malignant pleural effusion, and it can improve their quality of life (QOL). 順鉑聯(lián)合胸腺五肽治療惡性胸腔積液有確切療效,明顯提高化療藥物敏感性,進(jìn)而提高患者的生活質(zhì)量。
- Cisplatin and thymopentin were injected into thoracic cavity in trial group patients after all pleural fluid released out, but only cisplatin was injected in control group. 觀(guān)察組患者放盡胸水后經(jīng)胸腔內注入順鉑加胸腺五肽進(jìn)行治療,對照組患者放盡胸水后經(jīng)胸腔內注入順鉑進(jìn)行治療。
- Therefore, there's in need we should combine immune modulator, and anti-virus like polysaccharide, thymopentin or something, must combine anti-virus drugs. 因此,我們可以合并免疫調節藥物,例如云芝多糖,胸腺肽等,然后和抗病毒藥物一起使用。
- The pentapeptide Thymopentin (TP5) is the fragment of thymopoietin II(32-36) with basic sequence H-Arg-Lys-Asp-Val-Tyr-OH. It has the same biological activity as the thymopoietin II, which has the double-direction immunities to our bodies. 以H-Arg-Lys-Asp-Val-Tyr-OH 為序列的胸腺五肽(TP5)是胸腺生成素II(Thymopoietin II)中第32~36 位的氨基酸殘基片段,它保留了胸腺生成素II原有的生物活性,對機體的免疫系統具有雙向調節作用,現已作為藥物投放市場(chǎng)。
- HATU as the coupling reagent; TFA, p-methyl phenol, EDT and H2O (97:0.25:0.25:2.5) as the cleavage condition, the yield of thymopentin was 79.68% and the purity was 80.36% under 2 equiv. 反應結果胸腺五肽純度達80.;36%25;收率達79
- Teabag method was used to synthesize the peptide library of thymopentin with D-amino acids substituted by solid phase peptide synthesis (SPPS).Thirty-two peptides were synthesized. 利用組合化學(xué)技術(shù),采用簡(jiǎn)便的茶袋法固相合成制備胸腺五肽D型氨基酸取代類(lèi)似物肽庫,共合成32條肽。
- Conclusions There are some surely therapeutic effect for cisplatin combination with thymopentin on patients with malignant pleural effusion, and it can improve their quality of life (QOL). 結論順鉑聯(lián)合胸腺五肽治療惡性胸腔積液有確切療效,明顯提高化療藥物敏感性,進(jìn)而提高患者的生活質(zhì)量。
- thymopentin continuous release microspheres 胸腺五肽長(cháng)效微球
- Keywords microwave;cleavage;thymopentin;peptide resin; 微波;切割;胸腺五肽;肽樹(shù)脂;
- SEPARATION OF SOLID PHASE SYNTHESIS THYMOPENTIN USING ION-EXCHANGE METHOD 離子交換法分離固相合成胸腺五肽