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- opiate receptor agonist 鴉片受體拮抗劑
- The M receptor agonist pilocarpine was similar to the effects of ACh. M受體激動(dòng)劑毛果蕓香堿能產(chǎn)生與ACh相似的效應。
- BACKGROUND: As unspecific antagonist of opiate receptor, naloxone is widely used for multiple diseases which are related with abnormal release of endogenous opium. 背景:納洛酮作為阿片受體的非特異性拮抗劑,已被用于治療內源性阿片類(lèi)物質(zhì)異常釋放有關(guān)的多種疾病。
- Objective To investigate the effect of doparnine receptor agonist piribedil on dopamine transporter. 目的研究常用抗帕金森藥多巴胺受體激動(dòng)劑吡貝地爾(舒達)腦多巴胺轉運體的影響。
- Clinical treatment of PD includes dopamine replacement such as L-DOPA and D_2 dopamine receptor agonist. 目前臨床仍以替代治療為主,左旋多巴和D_2受體激動(dòng)劑能改善PD癥狀,但不能阻制疾病發(fā)展,這使人們對PD治療的認識由單純替代療法逐漸轉向保護中腦DA能神經(jīng)元。
- The presence of opiate receptors in .these neurons was identified. 2.;電刺激韁核可以使藍斑細胞的自發(fā)放電頻率增高。
- Rotigotine is a non-ergolinic dopamine receptor agonist available as a patch for once-daily use. 羅替戈汀是現有非二氫麥角堿多巴胺受體激動(dòng)劑中可作為每日一次使用的輔助藥物。
- Rotigotine is a non-ergolinic dopamine receptor agonist aailable as a patch for once-daily use. 羅替戈汀是現有非二氫麥角堿多巴胺受體激動(dòng)劑中可作為每日一次使用的輔助藥物。
- The citrated whole blood is tested at the basal and TRAP (Thrombin Receptor Agonist Peptide) activated states. 檸檬酸化的健康的血被測試在基礎并且捕捉(凝血酶感受器官收縮筋肽)被激活的狀態(tài)。
- A brief discussion is also given about the pr ospects of nicotinic receptor agonist used as non-opiate analgesics. 從地棘蛙素全合成研究、類(lèi)似物制備、藥理學(xué)行為和構效關(guān)系等幾方面介紹了國際上研究的熱點(diǎn),并對今后的研究動(dòng)向進(jìn)行了討論。
- The effects of receptor agonist and antagonist on hypnotic activity of melatonin were studied in the paper. 觀(guān)察不同受體激動(dòng)劑或拮抗劑對褪黑素催眠作用的影響。
- Objective: To study the protecting effect of delayed preconditioning with A1 selective adenosine receptor agonist in donor heart preservation. 目的:探討腺苷A1受體激動(dòng)劑延遲預處理對大鼠心臟的保護效果。
- The competition curves of inverse BDZ receptor agonist DMCM was illustrated in a biphasic way by a computer model of two sites. 反相激動(dòng)劑DMCM競爭結合曲線(xiàn)亦具有雙位點(diǎn)結合特性。
- Endorphins, a known substances produced in brains is an opioid receptor agonist which the brain produce in the presence of pain stimulus. 如果你一連幾天、一天幾次進(jìn)行實(shí)驗:誘發(fā)某人身感疼痛,再用嗎啡為他止疼,到最后一天,悄悄用鹽水取代嗎啡,你會(huì )發(fā)現,此時(shí)鹽水也能止痛。
- As a high-selective 5-HT1D receptor agonist, sumatriptan is mainly used as an emergency medicine in the treatment of migraine and cluster headache. 舒馬曲坦為具有高度選擇性的5-HT1D受體激動(dòng)劑,主要用作偏頭痛和叢集性頭痛發(fā)作的急救藥。
- Morphine binds strongly to opiate receptors in the brain to produce analgesia.In vitro studies on opiate receptors show that the quaternary salt of morphine also binds strongly. 嗎啡通過(guò)與大腦中的阿片受體緊密粘合產(chǎn)生止痛作用,在體外研究中,阿片受體與嗎啡的季鹽也有強力的粘合作用。
- The same question had arisen in the 1970s about morphine, a compound isolated from the poppy and found to bind to so-called opiate receptors in the brain. 相同的問(wèn)題于1970年代也出現過(guò),起因是從罌粟當中提煉出來(lái)的某個(gè)化合物,可與腦中所謂的鴉片受體結合。
- "Our findings suggest that elevated opiate receptors in the ventral striatum could be a biologic link between personality traits and dependence risk," they write. 參與者接著(zhù)接受心理測驗,以確認人格特性,包括尋求新穎事務(wù)、避免傷害、報酬依賴(lài)與持續情形。
- Any of a group of peptide hormones that bind to opiate receptors and are found mainly in the brain. Endorphins reduce the sensation of pain and affect emotions. 多肽,內啡肽指將麻醉傳感器聯(lián)結在一起的任一肽激素群,主要存在大腦中,內啡肽可緩解痛感并影響情緒
- Our results demonstrated for the first time that Spd, the dopamine D1 receptor agonist -D2 receptor antagonist, decreased the reinforcing efficacy of cocaine. 我們的研究首次發(fā)現,多巴胺D1受體激動(dòng)- D2受體拮抗劑左旋千金藤啶堿降低可卡因的獎賞效應;