Methods Starting with 3-fluorophenyl isocyanate and(R)-epichlorohydrin, linezolid was synthesized through cyclization, substitution, acylation, bromination, and condensation.

 
  • 方法以(R)-環(huán)氧氯丙烷和間氟苯基異氰酸酯為起始原料,經(jīng)環(huán)化、疊氮化、還原、?;?、溴代、縮合反應得到利奈唑酮。
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