Levocetirizine Dihydrochloride was prepared from benzoyl chloride by acidylation,hydrogenation,cyclization with an overall yield of 8.05%.

 
  • 以苯甲酰氯為原料;經(jīng)?;?;還原;環(huán)合等反應合成左旋西替利嗪鹽酸鹽;反應總收率為8.;05%25。
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