L-Asp6-Ibuprofen was prepared by mixture anhydrides methods and DCC/HOBt methods.The benzyl group of the product was deprotected by catalytic hydrogenation.

 
  • 方法使用混合酸酐法制備L-天冬氨酸六肽,分別用混合酸酐法和DCC法連接布洛芬,氫化還原得產(chǎn)物。
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